nib Malate≥99%341031-54-7100mg,500mg,1g无细胞VEGFR2 (Flk-1)80 nMPDGFRβ2 nML125046Lenalidomide≥99%191732-72-650mg,250mg,1g,5gPBMCsTNF-α13 nMC126195Cabozantinib (XL184, BMS-907351)≥98%849217-68-15mg,10mg,50mg,100mg,250mg无细胞VEGFR20.035 nMc-Met1.3 nM Ret4 nMKit4.6 nMFlt-1/3/412 nM/11.3 nM/6 nMTie214.3 nMAXL7 nMP127550Ponatinib (AP24534)≥99%943319-70-810mg,50mg,250mg无细胞Abl0.37 nMPDGFRα1.1 nMVEGFR21.5 nMFGFR12.2 nMSrc5.4 nMK125585Ki20227≥98%623142-96-110mg,50mgKDR2 nMVEGFR-212 nMc-Kit451 nMPDGFRβ217 nMA129732Axitinib≥99%319460-85-010mg,50mg,250mg,1g猪主动脉内皮细胞VEGFR10.1 nMVEGFR20.2 nMVEGFR30.1-0.3 nMPDGFRβ1.6 nMc-Kit1.7 nMF127011Foretinib (GSK1363089)≥98%849217-64-75mg,25mg,100mg无细胞Met0.4 nMKDR0.9 nMN129725Nintedanib (BIBF 1120)≥98%656247-17-55mg,10mg,25mg,50mg,100mg,500mg无细胞VEGFR134 nMVEGFR213 nMVEGFR313 nMFGFR169 nMFGFR237 nMFGFR3108 nMPDGFRα59 nMPDGFRβ65 nMV125180Vandetanib (ZD6474)≥99%443913-73-325mg,100mg,500mg无细胞VEGFR240 nMVEGFR3110 nMEGFR500 nMR127804Regorafenib (BAY 73-4506)≥99%755037-03-75mg,10mg,25mg,100mg无细胞VEGFR113 nMVEGFR24.2 nMVEGFR346 nMPDGFR-β22 nMKit7 nMRET1.5 nMRaf-12.5 nMP129722Pazopanib HCl (GW786034 HCl)≥98%635702-64-625mg,100mg,250mg,1g无细胞VEGFR110 nMVEGFR230 nMVEGFR347 nMPDGFR84 nMFGFR74 nMc-Kit140 nMc-fms146 nMC125911Cediranib≥98%288383-20-010mg,50mgVEGFR(KDR)<1 nMFlt1/45 nM/≤3 nMP125865PD173074≥99%219580-11-75mg,10mg,50mgFGFR125 nMVEGFR2100-200 nMD126778Dovitinib (TKI-258, CHIR-258)≥99%405169-16-610mg,50mg,250mg无细胞FLT31 nMc-Kit2 nML126993Linifanib (ABT-869)≥99%796967-16-35mg,10mg,50mgKDR4 nMCSF-1R3 nMFlt-1/33 nM/4 nMPDGFRβ66 nMV125857Vatalanib (PTK787) 2HCl≥99%212141-51-010mg,50mg无细胞VEGFR2/KDR37 nMR127906RAF265 (CHIR-265)≥98%927880-90-81mg,5mg,10mg,50mgVEGFR230 nMB-Raf3-60 nMT126012Tivozanib (AV-951)≥98%475108-18-05mg,25mg,100mgVEGFR10.21 nMVEGFR20.16 nMVEGFR30.24 nMM129736Motesanib Diphosphate (AMG-706)≥98%857876-30-35mg,10mg,50mgVEGFR12 nMVEGFR23 nMVEGFR36 nML125518Lenvatinib (E7080)≥99%417716-92-85mg,10mg,50mg,100mgVEGFR2(KDR)4 nMVEGFR3(Flt-4)5.2 nMB127317Brivanib (BMS-540215)≥98%649735-46-65mg,10mg,50mg VEGFR225 nMM127064MGCD-265≥98%875337-44-31mg,5mg,10mg,50mgc-Met1 nMVEGFR1/2/33 nM/3 nM/4 nMA126830AEE788 (NVP-AEE788)≥97%497839-62-05mg,25mg,100mgEGFR2 nMHER2/ErbB26 nME126318ENMD-2076≥99%934353-76-15mg,10mg,50mgAurora A14 nMFlt31.86 nMO126155OSI-930≥99%728033-96-31mg,5mg,25mg,50mgKit80 nMKDR9 nMCSF-1R15 nMC126929CYC116≥99%693228-63-61mg,10mg,50mgAurora A8.0 nMAurora B9.2 nMVEGFR244 nMK125876Ki8751≥98%228559-41-95mg,25mg,100mg VEGFR20.9 nMT129747Telatinib≥99%332012-40-51mg,5mg,10mg,50mgVEGFR2/36 nM/4 nMc-Kit1 nMPDGFRα15 nMP126419PP121≥98%1092788-83-410mg,50mgPDGFR2 nMHck8 nMmTOR10 nMVEGFR212 nMSrc14 nMAbl18 nMDNA-PK60 nMP125184Pazopanib≥99%444731-52-625mg,100mg,500mgGFR110 nMVEGFR230 nMVEGFR347 nMPDGFR84 nMFGFR74 nMc-Kit140 nMc-Fms/CSF1R146 nMK125907KRN-633≥97%286370-15-85mg,25mg,100mgVEGFR1170 nMVEGFR2160 nMVEGFR3125 nMS126571SAR131675≥99%1433953-83-31mg,10mg,50mg VEGFR323 nM12 nMB129768BMS-794833≥99%1174046-72-01mg,5mg,10mg,50mgMet1.7 nMVEGFR215 nMS125098Sorafenib≥99%284461-73-0250mg,1g无细胞Raf-16 nMB-Raf22 nM